Structural Biology

Visualize Success with Arctoris’ Advanced Structural Biology Solutions. Capabilities Overview

Capabilities Overview 

Arctoris accelerates your drug discovery by providing detailed structural insights into your targets and compounds. Our expert team and state-of-the-art technologies enable high-throughput co-crystallization, structural determination, and modeling. By elucidating binding modes and conformational changes, we empower you to implement rational, structure-guided drug design, enhancing the efficiency and success rate of your lead optimization efforts.

Key Features and Value

High-Throughput Crystallography: Process over 300 ligands efficiently for structural analysis.

Expert Modeling: Leverage our expertise to interpret structures and guide design.

Integrated Workflow: Combine structural data with biochemical and biophysical insights.

Rational Design: Utilize structural information to optimize potency and selectivity.

AI/ML Empowered: Generate structural datasets ideal for computational modeling.

Key Capabilities

Protein crystallization and co-crystallization with ligands

X-ray crystallography and structure determination

Cryo-electron microscopy for complex structures

Computational modeling and docking studies

Structural analysis of protein-ligand interactions

Integration with medicinal chemistry for design iterations

Data management and visualization tools

Validation Data

High Throughput: Established co-crystallization platforms for multiple targets.

Structural Success: Solved over 200 protein-ligand complex structures.

Potency Improvement: Enabled optimization improving compound potency by 10-fold.

Efficiency Gains: Accelerated lead optimization timelines by up to 30%.

Informed Decisions: Delivered structural insights supporting TMP achievement.